WebNov 25, 2024 · In this study, we explore the use of biolayer interferometry (BLI) as a tool for rapidly screening natural product sources for DNA targeting small molecules. ... or protein-DNA/RNA [33, 34] binding events, it has also been shown to be an excellent screening tool for small molecule interactions [30, 35, 36]. Here, we show for the first … WebOct 29, 2024 · Aptamers are functional single-stranded DNA or RNA oligo ... with a high KD of 0.93 nM 10 by SELEX and Biolayer interferometry ... D. J. Small-molecule interaction with a five-guanine-tract G ...
Biosensor-based small molecule fragment screening with …
WebFeb 2, 2024 · Biolayer interferometry (BLI) is a widely utilized technique for determining macromolecular interaction dynamics in real time. Using changes in the interference … WebMar 30, 2024 · Biolayer interferometry (BLI) and circular dichroism (CD) spectroscopy were used to investigate the interaction between previously reported i-motif DNA (i-DNA) ligands and folded or unfolded i-DNA in acidic (pH 5.5) and near-neutral (pH 6.5) conditions. We observed that although several ligands, in particula iron dream muscle pharm
Sougata Dey, Ph.D. - Lecturer - Texas A&M University
Web• Do not overload the immobilized molecule. • The same well containing buffer should be used for the baseline and dissociation phase, assuming inter-step correction is performed. • For small molecule work, use Super-Streptavidin sensors and quench with biocytin (biotinyl-lysine at 10 µg/mL). WebOct 11, 2024 · Introduction. RNA has diverse cellular functions and thus is an important target for small molecule chemical probes and lead therapeutics. 1, 2 The most exploited RNA targets for small molecules are three-dimensionally folded riboswitches 3 and ribosomes. 4, 5 Both are bacterial in origin, and small molecules that target these … WebLacI-DNA binding assayed with filter binding. The filter binding assay was used to monitor LacI binding to (a) lacO 1, (b) lacO 2, and (c) lacO 3 in the absence ( ) and presence ( ) of 1 mM IPTG. In these experiments, DNA concentration was fixed at 3 × 10 −12 M. The solid line represents the best fit of Equation (1) and the values reported in Table 2 are the … iron dream meaning